Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T8548 |
Metoprine
|
Histone Methyltransferase; Antifolate; Histamine Receptor | Cell Cycle/Checkpoint; Chromatin/Epigenetic; GPCR/G Protein; Immunology/Inflammation; Neuroscience |
Metoprine 是一种有效的组胺 N-甲基转移酶抑制剂,具有抗肿瘤活性。它是一种二氨基嘧啶衍生物,可以透过血脑屏障,并通过抑制 HMT 增加脑组胺水平。 |